Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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76
Tocris Bioscience™ TM 38837
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Highly potent CB1 inverse agonist; peripherally restricted
77
Tocris Bioscience™ JNJ 39758979 Dihydrochloride
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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High affinity and selective histamine H4 antagonist; orally bioavailable
| Purity | 98% |
|---|---|
| Chemical Name or Material | 4-[(3R)-3-Amino-1-pyrrolidinyl]-6-(1-methylethyl)-2-pyridinamine dihydrochloride |
| Recommended Storage | Desiccate at Room Temperature |
| Molecular Formula | C11H19N5.2HCl |
| Formula Weight | 294.22 |
78
Tocris Bioscience™ Phototrexate
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Photoswitchable inhibitor of human dihydrofolate reductase
79
Tocris Bioscience™ MS 154
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective cereblon-recruiting Degrader (PROTAC™) of mutant EGFR
80
Tocris Bioscience™ Thalidomide 5'-amine-alkylC6-amine
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Cereblon ligand with alkyl linker and terminal amine for onward chemistry
81
Tocris Bioscience™ Pomalidomide 4'-PEG5-amine
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Cereblon ligand with PEG linker and terminal amine for onward chemistry
82
Tocris Bioscience™ Squarunkin A Hydrochloride
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Small and Specialty Supplier Partner
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UNC119 chaperone-cargo interaction inhibitor; disrupts Src activation
| Purity | 98% |
|---|---|
| Chemical Name or Material | Ethyl 4-((3,4-dioxo-2-((2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)ethyl)amino)cyclobut-1-en-1-yl)amino)piperidine-1-carboxylate hydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C25H32F3N5O4.HCl |
| Formula Weight | 560.01 |
83
Tocris Bioscience™ PARPi-FL
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent fluorescent PARP inhibitor
84
Tocris Bioscience™ BDY FL, SE
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Small and Specialty Supplier Partner
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Green BDY (BODIPY™ or boron-dipyrromethene) fluorescent dye for the labeling of amines; supplied as NHS ester
85
Tocris Bioscience™ AZ 5704
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective ATM kinase inhibitor; orally bioavailable
| CAS | 1941214-06-7 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 7-Fluoro-6-[6-(methoxymethyl)-3-pyridinyl]-4-[[(1S)-1-(1-methyl-1H-pyrazol-3-yl)ethyl]amino]-3-quinolinecarboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C23H23FN6O2 |
| Formula Weight | 434.47 |
86
Tocris Bioscience™ A 410099.1 amide-PEG3-amine
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Small and Specialty Supplier Partner
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Small and Specialty Supplier Partner
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IAP ligand with PEG linker and terminal amine for onward chemistry
87
Tocris Bioscience™ BAY 805
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Potent and selective inhibitor of USP21; also NF-κB activator
| Target | Deubiquitinating Enzyme Inhibitors |
|---|---|
| CAS | 2925481-88-3 |
| Purity | 0.98 |
| Chemical Name or Material | N-[(1R)-1-[[[5-[(4-Cyanophenyl)methyl]-1,3,4-thiadiazol-2-yl]amino]carbonyl]-3-methylbutyl]-1-(trifluoromethyl)cyclohexanecarboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C24H28F3N5O2S |
88
Tocris Bioscience™ Dynarrestin
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Small and Specialty Supplier Partner
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Dynein inhibitor
89
Tocris Bioscience™ PSEM 308 hydrochloride
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PSAML141F-GlyR and PSAML141F,Y115F-5-HT3 chimeric ion channel agonist
| Target | Pharmacologically Selective Effector Molecules/PSEM |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 5-Methyl-5,8,9,10,11 A,12-hexahydro-4 H-8,11-ethanopyrido[3 ',2 ':3,4 ]diazepino[6,7,1-hi]indole hydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C17H21N3.HCl |
| Formula Weight | 303.83 |
90
Tocris Bioscience™ CHS 828
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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NAMPT inhibitor; active in vivo and cytotoxic
| CAS | 200484-11-3 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | N-[6-(4-Chlorophenoxy)hexyl]-N'-cyano-N''-4-pyridinylguanidine |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H22ClN5O |
| Formula Weight | 371.86 |